| 1. |
Hirose, Yuya; Shindo, Naoya; Mori, Makiko; Onitsuka, Satsuki; Isogai, Hikaru; Hamada, Rui; Hiramoto, Tadanari; Ochi, Jinta; Takahashi, Daisuke; Ueda, Tadashi; Caaveiro, Jose M. M.; Yoshida, Yuya; Ohdo, Shigehiro; Matsunaga, Naoya; Toba, Shinsuke; Sasaki, Michihito; Orba, Yasuko; Sawa, Hirofumi; Sato, Akihiko; Kawanishi, Eiji; Ojida, Akio, Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for Severe Acute Respiratory Syndrome Coronavirus 2 3CL Protease, Journal of Medicinal Chemistry, https://doi.org/10.1021/acs.jmedchem.2c01081, 65, 20, 13852-13865, 2022.10. |
| 2. |
Yamane, Daiki; Onitsuka, Satsuki; Re, Suyong; Isogai, Hikaru; Hamada, Rui; Hiramoto, Tadanari; Kawanishi, Eiji; Mizuguchi, Kenji; Shindo, Naoya; Ojida, Akio, Selective covalent targeting of SARS-CoV-2 main protease by enantiopure chlorofluoroacetamide, CHEMICAL SCIENCE, 10.1039/d1sc06596c, 13, 10, 3027-3034, 2022.03. |
| 3. |
Kumagai, Shinji; Sawamoto, Hiroaki; Takegawa-Araki, Tomo; Arai, Yuki; Yamakoshi, Shuhei; Yamada, Katsuya; Ohta, Tetsuya; Kawanishi, Eiji; Horie, Naohhiro; Yamaguchi, Takao; Obika, Satoshi, Synthesis and properties of GuNA purine/pyrimidine nucleosides and oligonucleotides, ORGANIC & BIOMOLECULAR CHEMISTRY, 10.1039/d0ob01970d, 18, 46, 9461-9472, 2020.12. |
| 4. |
Koizumi, Yuuki; Tanaka, Yoshihito; Matsumura, Takehiko; Kadoh, Yoichi; Miyoshi, Haruko; Hongu, Mitsuya; Takedomi, Kei; Kotera, Jun; Sasaki, Takashi; Taniguchi, Hiroyuki; Watanabe, Yumi; Takakuwa, Misae; Kojima, Koki; Baba, Nobuyuki; Nakamura, Itsuko; Kawanishi, Eiji, Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety, Bioorganic & Medicinal Chemistry, 10.1016/j.bmc.2019.06.021, 27, 15, 3440-3450, 2019.08. |
| 5. |
Yamagami, Takafumi; Kobayashi, Ryo; Moriyama, Noriaki; Horiuchi, Hideki; Toyofuku, Eiji; Kadoh, Yoichi; Kawanishi, Eiji; Izumoto, Shinichi; Hiramatsu, Hajime; Nanjo, Takehiro; Sugino, Masuhiro; Utsugi, Masayuki; Moritani, Yasunori, Scalable Process Design for a PDE10A Inhibitor Consisting of Pyrazolopyrimidine and Quinoxaline as Key Units, Organic Process Research & Development, 10.1021/acs.oprd.9b00068, 23, 4, 578-587, 2019.04. |
| 6. |
Sawamoto, Hiroaki; Arai, Yuuki; Yamakoshi, Shuhei; Obika, Satoshi; Kawanishi, Eiji, Synthetic Method for 2 '-Amino-LNA Bearing Any of the Four Nucleobases via a Transglycosylation Reaction, Organic Letters, 10.1021/acs.orglett.8b00476, 20, 7, 1928-1931, 2018.04. |
| 7. |
Kadoh, Yoichi; Miyoshi, Haruko; Matsumura, Takehiko; Tanaka, Yoshihito; Hongu, Mitsuya; Kimura, Mayumi; Takedomi, Kei; Omori, Kenji; Kotera, Jun; Sasaki, Takashi; Kobayashi, Tamaki; Taniguchi, Hiroyuki; Watanabe, Yumi; Kojima, Koki; Sakamoto, Toshiaki; Himiyama, Toshiyuki; Kawanishi, Eiji, Discovery of 2-[(E)-2-(7-Fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin-1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine Hydrochloride as a Highly Selective PDE10A Inhibitor, Chemical & Pharmaceutical Bulletin, 10.1248/cpb.c17-00783, 66, 3, 243-250, 2018.03. |
| 8. |
Yamakoshi, Shuhei; Okamoto, Masako; Sawamoto, Hiroaki; Arai, Yuuki; Kawanishi, Eiji; Sasaki, Michiko; Takeda, Kei, Computation-Assisted Disconnection Approach for the Synthesis of Neoantimycins, 15-Membered Macrocyclic Depsipeptides, Current Organic Synthesis, 10.2174/1570179413666160624105401, 14, 2, 299-308, 2017.02. |
| 9. |
Plisson, Christophe; Weinzimmer, David; Jakobsen, Steen; Natesan, Sridhar; Salinas, Cristian; Lin, Shu-Fei; Labaree, David; Zheng, Ming-Qiang; Nabulsi, Nabeel; Marques, Tiago Reis; Kapur, Shitij; Kawanishi, Eiji; Saijo, Takeaki; Gunn, Roger N.; Carson, Richard E.; Rabiner, Eugenii A., Phosphodiesterase 10A PET Radioligand Development Program: From Pig to Human, JOURNAL OF NUCLEAR MEDICINE, 10.2967/jnumed.113.131409, 55, 4, 595-601, 2014.04. |
| 10. |
Yamakoshi, Shuhei; Kawanishi, Eiji, First total synthesis of prunustatin A, Tetrahedron Letters, 10.1016/j.tetlet.2013.12.106, 55, 6, 1175-1177, 2014.02. |
| 11. |
Yamamoto, Yasuo; Kawanishi, Eiji; Koga, Yuichi; Sakamaki, Shigeki; Sakamoto, Toshiaki; Ueta, Kiichiro; Matsushita, Yasuaki; Kuriyama, Chiaki; Tsuda-Tsukimoto, Minoru; Nomura, Sumihiro, N-glucosides as human sodium-dependent glucose cotransporter 2 (hSGLT2) inhibitors, Bioorganic & Medicinal Chemistry, 10.1016/j.bmcl.2013.08.042, 23, 20, 5641-5645, 2013.10. |
| 12. |
Koga, Yuichi; Sakamaki, Shigeki; Hongu, Mitsuya; Kawanishi, Eiji; Sakamoto, Toshiaki; Yamamoto, Yasuo; Kimata, Hirotaka; Nakayama, Keiko; Kuriyama, Chiaki; Matsushita, Yasuaki; Ueta, Kiichiro; Tsuda-Tsukimoto, Minoru; Nomura, Sumihiro, C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors, Bioorganic & Medicinal Chemistry, 10.1016/j.bmc.2013.05.048, 21, 17, 5561-5572, 2013.09. |
| 13. |
Sakamaki, Shigeki; Kawanishi, Eiji; Koga, Yuichi; Yamamoto, Yasuo; Kuriyama, Chiaki; Matsushita, Yasuaki; Ueta, Kiichiro; Nomura, Sumihiro, Synthesis and biological evaluation of thiophene-C-glucosides as sodium-dependent glucose Co-transporter 2 inhibitors, Chemical & Pharmaceutical Bulletin, 10.1248/cpb.c13-00407, 61, 10, 1037-1043, 2013.08. |
| 14. |
Plisson, Christophe; Salinas, Cristian; Weinzimmer, David; Labaree, David; Lin Shu-Fei; Zheng Ming-Qiang; Nabulsi, Nabeel; Jakobsen, Steen; Kawanishi, Eiji; Saijo, Takeaki; Carson, Richard; Gunn, Roger; Rabiner, Eugenii, Radiosynthesis and in vivo evaluation in the pig and baboon of candidate phosphodiesterase 10A PET radioligands. Comparison with [C-11]MP-10., JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 56, S301-S301, 2013.05. |
| 15. |
Sakamaki, Shigeki; Kawanishi, Eiji; Nomura, Sumihiro; Ishikawa, Tsutomu, Aryl-beta-C-glucosidation using glucal boronate: application to the synthesis of tri-O-methylnorbergenin, Tetrahedron, 10.1016/j.tet.2012.05.035, 68, 29, 5744-5753, 2012.07. |
| 16. |
Plisson, Christophe; Salinas, Cristian; Weinzimmer, David; Labaree, David; Lin, Shu-Fei; Ding, Yu-Shin; Jakobsen, Steen; Smith, Paul W.; Kawanishi, Eiji; Carson, Richard E.; Gunn, Roger N.; Rabiner, Eugenii A., Radiosynthesis and in vivo evaluation of [C-11]MP-10 as a positron emission tomography radioligand for phosphodiesterase 10A, NUCLEAR MEDICINE AND BIOLOGY, 10.1016/j.nucmedbio.2011.02.005, 38, 6, 875-884, 2011.08. |
| 17. |
Nomura, Sumihiro; Sakamaki, Shigeki; Hongu, Mitsuya; Kawanishi, Eiji; Koga, Yuichi; Sakamoto, Toshiaki; Yamamoto, Yasuo; Ueta, Kiichiro; Kimata, Hirotaka; Nakayama, Keiko; Tsuda-Tsukimoto, Minoru, Discovery of Canagliflozin, a Novel C-Glucoside with Thiophene Ring, as Sodium-Dependent Glucose Cotransporter 2 Inhibitor for the Treatment of Type 2 Diabetes Mellitus, Jornal of Medicinal Chemistry, 10.1021/jm100332n, 53, 17, 6355-6360, 2010.09. |
| 18. |
Sasaki, Michiko; Kawanishi, Eiji; Shirakawa, Yuri; Kawahata, Masatoshi; Masu, Hyuma; Yamaguchi, Kentaro; Takeda, Kei, Chirality transfer from epoxide to carbanion: Base-induced alkylation of O-carbamoyl cyanohydrins of beta-silyl-alpha,beta-epoxy aldehyde, European Jornal of Organic Chemistry, 10.1002/ejoc.200800300, 18, 3061-3064, 2008.06. |
| 19. |
Sasaki, Michiko; Kawanishi, Eiji; Nakai, Yoshio; Matsumoto, Tatsuya; Yamaguchi, Kentaro; Takeda, Kei, Tandem Base-Promoted Ring-Opening/Brook Rearrangement/Allylic Alkylation of O-Silyl Cyanohydrins of β-Silyl-α,β-epoxyaldehyde: Scope and Mechanism, Journal of Organic Chemistry, 10.1021/jo0352934, 68, 24, 9330-9339, 2003.11. |
| 20. |
Takeda, Kei; Kawanishi, Eiji; Sasaki, Michiko; Takahashi, Yuji; Yamaguchi, Kentaro, Tandem Base-Promoted Ring Opening/Brook Rearrangement/Allylic Alkylation of O-Silyl Cyanohydrins of β-Silyl-α,β-epoxyaldehydes, Organic Letters, 10.1021/ol025738v, 4, 9, 1151-1154, 2002.05. |
| 21. |
Kawanishi, Eiji; Higuchi, Kyoichi; Ishida, Akihiko, Synthesis of N,N'-unsymmetrical diacylcystines and cystine-containing dipeptides, Heterocycles, 10.3987/COM-99-S52, 52, 1, 425-442, ISSN:0385-5414, 2000.01. |
| 22. |
Takeda, Kei; Kawanishi, Eiji; Nakamura, Hitoshi; Yoshii, Eiichi, Total synthesis of tetronolide, the aglycon of tetrocarcins, Tetrahedron Letters, 10.1016/S0040-4039(00)93498-1, 32, 37, 4925-4928, 1991.09. |
